Target Disease Drug_index Drug ADRB2 Chronic Obstructive Pulmonary Disease 1 albuterol [Beta-2 adrenergic receptor agonist], albuterol sulfate [Beta-2 adrenergic receptor agonist], arformoterol tartrate [Beta-2 adrenergic receptor agonist], formoterol fumarate [Beta-2 adrenergic receptor agonist], indacaterol maleate [Beta-2 adrenergic receptor agonist], olodaterol hydrochloride [Beta-2 adrenergic receptor agonist], salmeterol xinafoate [Beta-2 adrenergic receptor agonist], vilanterol trifenatate [Beta-2 adrenergic receptor agonist] ADRB2 Asthma 2 albuterol [Beta-2 adrenergic receptor agonist], albuterol sulfate [Beta-2 adrenergic receptor agonist], formoterol fumarate [Beta-2 adrenergic receptor agonist], levalbuterol hydrochloride [Beta-2 adrenergic receptor agonist], metaproterenol sulfate [Beta-2 adrenergic receptor agonist], pirbuterol acetate [Beta-2 adrenergic receptor agonist], salmeterol xinafoate [Beta-2 adrenergic receptor agonist], terbutaline sulfate [Beta-2 adrenergic receptor agonist], vilanterol trifenatate [Beta-2 adrenergic receptor agonist] ADRB2 Bronchospasm 3 albuterol [Beta-2 adrenergic receptor agonist], albuterol sulfate [Beta-2 adrenergic receptor agonist], formoterol fumarate [Beta-2 adrenergic receptor agonist], salmeterol xinafoate [Beta-2 adrenergic receptor agonist], terbutaline sulfate [Beta-2 adrenergic receptor agonist] ADRB2 Airway Obstruction 4 albuterol [Beta-2 adrenergic receptor agonist], clenbuterol [Beta-2 adrenergic receptor agonist], rimiterol [Beta-2 adrenergic receptor agonist], tulobuterol [Beta-2 adrenergic receptor agonist] PDE4D Airway Obstruction 5 aminophylline [Phosphodiesterase 4 inhibitor], amlexanox [Phosphodiesterase 4 inhibitor], dyphylline [Phosphodiesterase 4 inhibitor], oxtriphylline [Phosphodiesterase 4 inhibitor], roflumilast [Phosphodiesterase 4 inhibitor], theophylline [Phosphodiesterase 4 inhibitor] PDE4D Asthma 6 aminophylline [Phosphodiesterase 4 inhibitor], theophylline [Phosphodiesterase 4 inhibitor] DRD2 Psychosis 7 amisulpride [Dopamine receptors; D2 & D3 antagonist], aripiprazole [Dopamine D2 receptor partial agonist], benperidol [Dopamine D2 receptor antagonist], brexpiprazole [Dopamine D2 receptor partial agonist], bromperidol [Dopamine D2 receptor antagonist], chlorpromazine [D2-like dopamine receptor antagonist], chlorprothixene [Dopamine D2 receptor antagonist], clozapine [Dopamine D2 receptor antagonist], droperidol [D2-like dopamine receptor antagonist], fluphenazine decanoate [Dopamine D2 receptor antagonist], fluphenazine enanthate [Dopamine D2 receptor antagonist], haloperidol [D2-like dopamine receptor inverse agonist], haloperidol decanoate [D2-like dopamine receptor inverse agonist], iloperidone [Dopamine D2 receptor antagonist], levomepromazine [D2-like dopamine receptor antagonist], loxapine [D2-like dopamine receptor antagonist], olanzapine [D2-like dopamine receptor antagonist], paliperidone [Dopamine D2 receptor antagonist], perphenazine [Dopamine D2 receptor antagonist], pimozide [Dopamine receptor antagonist], prochlorperazine [Dopamine D2 receptor antagonist], risperidone [Dopamine D2 receptor antagonist], sulpiride [Dopamine D2 receptor antagonist], thiothixene [Dopamine D2 receptor antagonist], triflupromazine [Dopamine D2 receptor antagonist] DRD2 Nausea And Vomiting 8 amisulpride [Dopamine receptors; D2 & D3 antagonist], chlorpromazine [D2-like dopamine receptor antagonist], droperidol [D2-like dopamine receptor antagonist], metoclopramide hydrochloride [Dopamine D2 receptor antagonist], perphenazine [Dopamine D2 receptor antagonist], prochlorperazine [Dopamine D2 receptor antagonist] DRD2 Post Operative Nausea And Vomiting 9 amisulpride [Dopamine receptors; D2 & D3 antagonist], droperidol [D2-like dopamine receptor antagonist], metoclopramide hydrochloride [Dopamine D2 receptor antagonist] CACNA1S Heart Failure 10 amlodipine benzoate [Voltage-gated L-type calcium channel blocker] CACNA1F Heart Failure 10 amlodipine benzoate [Voltage-gated L-type calcium channel blocker] CACNA1D Heart Failure 10 amlodipine benzoate [Voltage-gated L-type calcium channel blocker] CACNA1C Heart Failure 10 amlodipine benzoate [Voltage-gated L-type calcium channel blocker] CACNA1S Coronary Artery Disease 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Coronary Artery Disease 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Coronary Artery Disease 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Coronary Artery Disease 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Myocardial Infarction 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Myocardial Infarction 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Myocardial Infarction 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Myocardial Infarction 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Stroke 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Stroke 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Stroke 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Stroke 11 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Hypertension 12 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], levamlodipine maleate [Voltage-gated L-type calcium channel blocker], nicardipine hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Hypertension 12 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], levamlodipine maleate [Voltage-gated L-type calcium channel blocker], nicardipine hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Hypertension 12 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], levamlodipine maleate [Voltage-gated L-type calcium channel blocker], nicardipine hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Hypertension 12 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], levamlodipine maleate [Voltage-gated L-type calcium channel blocker], nicardipine hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1S Diabetes Mellitus 13 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Diabetes Mellitus 13 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Diabetes Mellitus 13 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Diabetes Mellitus 13 amlodipine benzoate [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1S Congestive Heart Failure 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Congestive Heart Failure 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Congestive Heart Failure 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Congestive Heart Failure 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Familial Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Familial Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Familial Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Familial Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Hypercholesterolemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Hyperlipidemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Hyperlipidemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Hyperlipidemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Hyperlipidemia 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Prinzmetal's Angina 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1F Prinzmetal's Angina 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1D Prinzmetal's Angina 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1C Prinzmetal's Angina 14 amlodipine besylate [Voltage-gated L-type calcium channel blocker] CACNA1S Angina Pectoris 15 amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Angina Pectoris 15 amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Angina Pectoris 15 amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Angina Pectoris 15 amlodipine besylate [Voltage-gated L-type calcium channel blocker], diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] DRD2 Unipolar Depression 16 amoxapine [Dopamine receptor antagonist], aripiprazole [Dopamine D2 receptor partial agonist], brexpiprazole [Dopamine D2 receptor partial agonist], olanzapine [D2-like dopamine receptor antagonist], quetiapine fumarate [Dopamine D2 receptor antagonist] DRD2 Parkinson's Disease 17 apomorphine hydrochloride [D2-like dopamine receptor agonist], bromocriptine mesylate [D2-like dopamine receptor agonist], cabergoline [Dopamine D2 receptor agonist], pramipexole dihydrochloride [D2-like dopamine receptor agonist], ropinirole hydrochloride [D2-like dopamine receptor agonist], rotigotine [D2-like dopamine receptor agonist] PDE4D Oral Ulcer 18 apremilast [Phosphodiesterase 4 inhibitor] PDE4D Psoriasis 18 apremilast [Phosphodiesterase 4 inhibitor] PDE4D Psoriatic Arthritis 18 apremilast [Phosphodiesterase 4 inhibitor] PDE4D Pustulosis Palmaris Et Plantaris 18 apremilast [Phosphodiesterase 4 inhibitor] ADRB2 Chronic Bronchitis 19 arformoterol tartrate [Beta-2 adrenergic receptor agonist], formoterol fumarate [Beta-2 adrenergic receptor agonist], indacaterol maleate [Beta-2 adrenergic receptor agonist], olodaterol hydrochloride [Beta-2 adrenergic receptor agonist], salmeterol xinafoate [Beta-2 adrenergic receptor agonist], vilanterol trifenatate [Beta-2 adrenergic receptor agonist] ADRB2 Emphysema 19 arformoterol tartrate [Beta-2 adrenergic receptor agonist], formoterol fumarate [Beta-2 adrenergic receptor agonist], indacaterol maleate [Beta-2 adrenergic receptor agonist], olodaterol hydrochloride [Beta-2 adrenergic receptor agonist], salmeterol xinafoate [Beta-2 adrenergic receptor agonist], vilanterol trifenatate [Beta-2 adrenergic receptor agonist] DRD2 Depressive Disorder 20 aripiprazole [Dopamine D2 receptor partial agonist] DRD2 Schizophrenia 21 aripiprazole [Dopamine D2 receptor partial agonist], aripiprazole lauroxil [Dopamine D2 receptor partial agonist], asenapine maleate [Dopamine D2 receptor antagonist], brexpiprazole [Dopamine D2 receptor partial agonist], cariprazine hydrochloride [Dopamine D2 receptor modulator], chlorpromazine [D2-like dopamine receptor antagonist], clozapine [Dopamine D2 receptor antagonist], haloperidol [D2-like dopamine receptor inverse agonist], haloperidol decanoate [D2-like dopamine receptor inverse agonist], haloperidol lactate [D2-like dopamine receptor inverse agonist], iloperidone [Dopamine D2 receptor antagonist], loxapine [D2-like dopamine receptor antagonist], lurasidone hydrochloride [Dopamine D2 receptor antagonist], molindone hydrochloride [Dopamine D2 receptor antagonist], olanzapine [D2-like dopamine receptor antagonist], olanzapine pamoate [D2-like dopamine receptor antagonist], paliperidone [Dopamine D2 receptor antagonist], paliperidone palmitate [Dopamine D2 receptor antagonist], perphenazine [Dopamine D2 receptor antagonist], prochlorperazine [Dopamine D2 receptor antagonist], quetiapine fumarate [Dopamine D2 receptor antagonist], risperidone [Dopamine D2 receptor antagonist], thiothixene [Dopamine D2 receptor antagonist], trifluoperazine hydrochloride [D2-like dopamine receptor antagonist], ziprasidone hydrochloride [Dopamine D2 receptor antagonist] DRD2 Bipolar I Disorder 22 aripiprazole [Dopamine D2 receptor partial agonist], aripiprazole lauroxil [Dopamine D2 receptor partial agonist], asenapine maleate [Dopamine D2 receptor antagonist], cariprazine hydrochloride [Dopamine D2 receptor modulator], loxapine [D2-like dopamine receptor antagonist], lurasidone hydrochloride [Dopamine D2 receptor antagonist], olanzapine [D2-like dopamine receptor antagonist], olanzapine pamoate [D2-like dopamine receptor antagonist], quetiapine fumarate [Dopamine D2 receptor antagonist], risperidone [Dopamine D2 receptor antagonist], ziprasidone hydrochloride [Dopamine D2 receptor antagonist] DRD2 Major Depressive Disorder 23 aripiprazole [Dopamine D2 receptor partial agonist], aripiprazole lauroxil [Dopamine D2 receptor partial agonist], brexpiprazole [Dopamine D2 receptor partial agonist], olanzapine [D2-like dopamine receptor antagonist], quetiapine fumarate [Dopamine D2 receptor antagonist] DRD2 Autism 24 aripiprazole [Dopamine D2 receptor partial agonist], aripiprazole lauroxil [Dopamine D2 receptor partial agonist], risperidone [Dopamine D2 receptor antagonist] DRD2 Bipolar Disorder 25 aripiprazole [Dopamine D2 receptor partial agonist], asenapine maleate [Dopamine D2 receptor antagonist], cariprazine hydrochloride [Dopamine D2 receptor modulator], lurasidone hydrochloride [Dopamine D2 receptor antagonist], olanzapine [D2-like dopamine receptor antagonist], quetiapine fumarate [Dopamine D2 receptor antagonist], risperidone [Dopamine D2 receptor antagonist], ziprasidone hydrochloride [Dopamine D2 receptor antagonist], ziprasidone mesylate [Dopamine D2 receptor antagonist] DRD2 Schizoaffective Disorder 26 aripiprazole [Dopamine D2 receptor partial agonist], brexpiprazole [Dopamine D2 receptor partial agonist], clozapine [Dopamine D2 receptor antagonist], haloperidol [D2-like dopamine receptor inverse agonist], olanzapine [D2-like dopamine receptor antagonist], paliperidone [Dopamine D2 receptor antagonist], paliperidone palmitate [Dopamine D2 receptor antagonist], risperidone [Dopamine D2 receptor antagonist] DRD2 Agitation 27 aripiprazole [Dopamine D2 receptor partial agonist], loxapine [D2-like dopamine receptor antagonist], olanzapine [D2-like dopamine receptor antagonist], olanzapine pamoate [D2-like dopamine receptor antagonist], ziprasidone hydrochloride [Dopamine D2 receptor antagonist] DRD2 Aggressive Behavior 28 aripiprazole [Dopamine D2 receptor partial agonist], risperidone [Dopamine D2 receptor antagonist] HTR2A Schizophrenia 29 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], aripiprazole lauroxil [Serotonin 2a (5-HT2a) receptor antagonist], asenapine maleate [Serotonin 2a (5-HT2a) receptor antagonist], brexpiprazole [Serotonin 2a (5-HT2a) receptor antagonist], chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist], clozapine [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol decanoate [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol lactate [Serotonin 2a (5-HT2a) receptor antagonist], iloperidone [Serotonin 2a (5-HT2a) receptor antagonist], loxapine [Serotonin 2a (5-HT2a) receptor antagonist], lurasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], molindone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine pamoate [Serotonin 2a (5-HT2a) receptor antagonist], paliperidone [Serotonin 2a (5-HT2a) receptor antagonist], paliperidone palmitate [Serotonin 2a (5-HT2a) receptor antagonist], quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist], thiothixene [Serotonin 2a (5-HT2a) receptor antagonist], trifluoperazine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Bipolar I Disorder 30 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], aripiprazole lauroxil [Serotonin 2a (5-HT2a) receptor antagonist], asenapine maleate [Serotonin 2a (5-HT2a) receptor antagonist], loxapine [Serotonin 2a (5-HT2a) receptor antagonist], lurasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine pamoate [Serotonin 2a (5-HT2a) receptor antagonist], quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist], ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Major Depressive Disorder 31 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], aripiprazole lauroxil [Serotonin 2a (5-HT2a) receptor antagonist], brexpiprazole [Serotonin 2a (5-HT2a) receptor antagonist], mirtazapine [Serotonin 2a (5-HT2a) receptor antagonist], nefazodone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist], trazodone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Autism 32 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], aripiprazole lauroxil [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Bipolar Disorder 33 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], asenapine maleate [Serotonin 2a (5-HT2a) receptor antagonist], lurasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist], ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], ziprasidone mesylate [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Psychosis 34 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], brexpiprazole [Serotonin 2a (5-HT2a) receptor antagonist], chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist], chlorprothixene [Serotonin 2a (5-HT2a) receptor antagonist], clothiapine [Serotonin 2 (5-HT2) receptor antagonist], clozapine [Serotonin 2a (5-HT2a) receptor antagonist], droperidol [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol decanoate [Serotonin 2a (5-HT2a) receptor antagonist], iloperidone [Serotonin 2a (5-HT2a) receptor antagonist], loxapine [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], paliperidone [Serotonin 2a (5-HT2a) receptor antagonist], pimavanserin tartrate [Serotonin 2a (5-HT2a) receptor inverse agonist], pimozide [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist], thiothixene [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Schizoaffective Disorder 35 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], brexpiprazole [Serotonin 2a (5-HT2a) receptor antagonist], clozapine [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], paliperidone [Serotonin 2a (5-HT2a) receptor antagonist], paliperidone palmitate [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Unipolar Depression 36 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], brexpiprazole [Serotonin 2a (5-HT2a) receptor antagonist], mirtazapine [Serotonin 2a (5-HT2a) receptor antagonist], nefazodone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist], trazodone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Agitation 37 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], loxapine [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine [Serotonin 2a (5-HT2a) receptor antagonist], olanzapine pamoate [Serotonin 2a (5-HT2a) receptor antagonist], ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Depressive Disorder 38 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], mirtazapine [Serotonin 2a (5-HT2a) receptor antagonist], trazodone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Aggressive Behavior 39 aripiprazole [Serotonin 2a (5-HT2a) receptor antagonist], risperidone [Serotonin 2a (5-HT2a) receptor antagonist] DRD2 Tourette Syndrome 40 aripiprazole lauroxil [Dopamine D2 receptor partial agonist], haloperidol [D2-like dopamine receptor inverse agonist], haloperidol decanoate [D2-like dopamine receptor inverse agonist], pimozide [Dopamine receptor antagonist] HTR2A Tourette Syndrome 41 aripiprazole lauroxil [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol decanoate [Serotonin 2a (5-HT2a) receptor antagonist], pimozide [Serotonin 2a (5-HT2a) receptor antagonist] PPARA Cardiovascular Disease 42 bezafibrate [Peroxisome proliferator-activated receptor agonist], choline fenofibrate [Peroxisome proliferator-activated receptor alpha agonist], ciprofibrate [Peroxisome proliferator-activated receptor alpha agonist], clofibrate [Peroxisome proliferator-activated receptor alpha agonist], fenofibrate [Peroxisome proliferator-activated receptor alpha agonist], gemfibrozil [Peroxisome proliferator-activated receptor alpha agonist] DRD2 Acromegaly 43 bromocriptine mesylate [D2-like dopamine receptor agonist] DRD2 Adenoma 43 bromocriptine mesylate [D2-like dopamine receptor agonist] DRD2 Hyperprolactinemia 43 bromocriptine mesylate [D2-like dopamine receptor agonist] DRD2 Hypogonadism 43 bromocriptine mesylate [D2-like dopamine receptor agonist] DRD2 Infertility 43 bromocriptine mesylate [D2-like dopamine receptor agonist] DRD2 Type Ii Diabetes Mellitus 43 bromocriptine mesylate [D2-like dopamine receptor agonist] ADRB2 Open-Angle Glaucoma 44 carteolol hydrochloride [Adrenergic receptor beta antagonist], timolol [Beta-2 adrenergic receptor antagonist], timolol maleate [Beta-2 adrenergic receptor antagonist] ADRB2 Heart Failure 45 carvedilol [Adrenergic receptor beta antagonist] ADRB2 Myocardial Infarction 46 carvedilol [Adrenergic receptor beta antagonist], carvedilol phosphate [Adrenergic receptor beta antagonist], nadolol [Beta-2 adrenergic receptor antagonist] ADRB2 Hypertension 47 carvedilol [Adrenergic receptor beta antagonist], carvedilol phosphate [Adrenergic receptor beta antagonist], nadolol [Beta-2 adrenergic receptor antagonist], nebivolol hydrochloride [Beta-2 adrenergic receptor antagonist], propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Cardiovascular Disease 48 carvedilol [Adrenergic receptor beta antagonist], celiprolol [Beta-2 adrenergic receptor partial agonist], nadolol [Beta-2 adrenergic receptor antagonist], pindolol [Beta-2 adrenergic receptor partial agonist], timolol [Beta-2 adrenergic receptor antagonist] ADRB2 Congestive Heart Failure 49 carvedilol [Adrenergic receptor beta antagonist], dobutamine hydrochloride [Beta-2 adrenergic receptor agonist], isoproterenol hydrochloride [Adrenergic receptor beta agonist] DRD2 Porphyria 50 chlorpromazine [D2-like dopamine receptor antagonist] DRD2 Mental Or Behavioural Disorder 51 chlorpromazine [D2-like dopamine receptor antagonist], fluphenazine decanoate [Dopamine D2 receptor antagonist], haloperidol decanoate [D2-like dopamine receptor inverse agonist], trifluoperazine hydrochloride [D2-like dopamine receptor antagonist] DRD2 Conduct Disorder 52 chlorpromazine [D2-like dopamine receptor antagonist], haloperidol [D2-like dopamine receptor inverse agonist], haloperidol decanoate [D2-like dopamine receptor inverse agonist] HTR2A Porphyria 53 chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Nausea And Vomiting 54 chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist], droperidol [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Conduct Disorder 55 chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol decanoate [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Mental Or Behavioural Disorder 56 chlorpromazine [Serotonin 2a (5-HT2a) receptor antagonist], haloperidol decanoate [Serotonin 2a (5-HT2a) receptor antagonist], trifluoperazine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] CACNA1S Vertigo 57 cinnarizine [Voltage-gated L-type calcium channel blocker] CACNA1F Vertigo 57 cinnarizine [Voltage-gated L-type calcium channel blocker] CACNA1D Vertigo 57 cinnarizine [Voltage-gated L-type calcium channel blocker] CACNA1C Vertigo 57 cinnarizine [Voltage-gated L-type calcium channel blocker] DRD2 Gastrointestinal Disease 58 clebopride [Dopamine D2 receptor antagonist], domperidone [Dopamine D2 receptor antagonist] CACNA1S Cardiovascular Disease 59 clevidipine [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nimodipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], nitrendipine [Voltage-gated L-type calcium channel blocker] CACNA1F Cardiovascular Disease 59 clevidipine [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nimodipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], nitrendipine [Voltage-gated L-type calcium channel blocker] CACNA1D Cardiovascular Disease 59 clevidipine [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nimodipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], nitrendipine [Voltage-gated L-type calcium channel blocker] CACNA1C Cardiovascular Disease 59 clevidipine [Voltage-gated L-type calcium channel blocker], felodipine [Voltage-gated L-type calcium channel blocker], isradipine [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker], nimodipine [Voltage-gated L-type calcium channel blocker], nisoldipine [Voltage-gated L-type calcium channel blocker], nitrendipine [Voltage-gated L-type calcium channel blocker] PDE4D Atopic Eczema 60 crisaborole [Phosphodiesterase 4 inhibitor] PDE4D Eczema 60 crisaborole [Phosphodiesterase 4 inhibitor] HTR2A Cerebral Palsy 61 cyclobenzaprine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Muscle Spasm 61 cyclobenzaprine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Myalgia 61 cyclobenzaprine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Spasticity 61 cyclobenzaprine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Spinal Cord Disease 61 cyclobenzaprine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] CACNA1S Syndromic Disease 62 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Syndromic Disease 62 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Syndromic Disease 62 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Syndromic Disease 62 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1S Atrial Fibrillation 63 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], dronedarone hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Atrial Fibrillation 63 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], dronedarone hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Atrial Fibrillation 63 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], dronedarone hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Atrial Fibrillation 63 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], dronedarone hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1S Coronary Vasospasm 64 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker] CACNA1F Coronary Vasospasm 64 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker] CACNA1D Coronary Vasospasm 64 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker] CACNA1C Coronary Vasospasm 64 diltiazem hydrochloride [Voltage-gated L-type calcium channel blocker], nifedipine [Voltage-gated L-type calcium channel blocker] HTR2A Post Operative Nausea And Vomiting 65 droperidol [Serotonin 2a (5-HT2a) receptor antagonist] DRD2 Cardiovascular Disease 66 ergoloid mesylates [Dopamine receptor agonist] PPARA Abnormal Circulating Lipid Concentration 67 fenofibrate [Peroxisome proliferator-activated receptor alpha agonist] PPARA Diabetes Mellitus 67 fenofibrate [Peroxisome proliferator-activated receptor alpha agonist] PPARA Hypothyroidism 67 fenofibrate [Peroxisome proliferator-activated receptor alpha agonist] PPARA Hypercholesterolemia 68 fenofibrate [Peroxisome proliferator-activated receptor alpha agonist], fenofibric acid [Peroxisome proliferator-activated receptor alpha agonist] PPARA Type Ii Diabetes Mellitus 68 fenofibrate [Peroxisome proliferator-activated receptor alpha agonist], fenofibric acid [Peroxisome proliferator-activated receptor alpha agonist] PDE4D Dysuria 69 flavoxate hydrochloride [Phosphodiesterase 4 inhibitor] PDE4D Prostatitis 69 flavoxate hydrochloride [Phosphodiesterase 4 inhibitor] PDE4D Urethritis 69 flavoxate hydrochloride [Phosphodiesterase 4 inhibitor] PDE4D Urinary Tract Infection 69 flavoxate hydrochloride [Phosphodiesterase 4 inhibitor] PPARA Abdominal Pain 70 gemfibrozil [Peroxisome proliferator-activated receptor alpha agonist] PPARA Coronary Artery Disease 70 gemfibrozil [Peroxisome proliferator-activated receptor alpha agonist] ADRB2 Glaucoma 71 levobunolol hydrochloride [Beta-2 adrenergic receptor antagonist], timolol [Beta-2 adrenergic receptor antagonist], timolol maleate [Beta-2 adrenergic receptor antagonist] DRD2 Anorexia 72 metoclopramide hydrochloride [Dopamine D2 receptor antagonist] DRD2 Gastroparesis 72 metoclopramide hydrochloride [Dopamine D2 receptor antagonist] DRD2 Kidney Failure 72 metoclopramide hydrochloride [Dopamine D2 receptor antagonist] DRD2 Vomiting 72 metoclopramide hydrochloride [Dopamine D2 receptor antagonist] HTR2A Insomnia 73 mirtazapine [Serotonin 2a (5-HT2a) receptor antagonist] ADRB2 Stroke 74 nadolol [Beta-2 adrenergic receptor antagonist], nebivolol hydrochloride [Beta-2 adrenergic receptor antagonist], propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Angina Pectoris 75 nadolol [Beta-2 adrenergic receptor antagonist], propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] OXTR Hemorrhage 76 oxytocin [Oxytocin receptor agonist] OXTR Uterine Inertia 76 oxytocin [Oxytocin receptor agonist] HTR2A Hallucinations 77 pimavanserin tartrate [Serotonin 2a (5-HT2a) receptor inverse agonist] HTR2A Parkinson's Disease 77 pimavanserin tartrate [Serotonin 2a (5-HT2a) receptor inverse agonist] DRD2 Restless Legs Syndrome 78 pramipexole dihydrochloride [D2-like dopamine receptor agonist], ropinirole hydrochloride [D2-like dopamine receptor agonist], rotigotine [D2-like dopamine receptor agonist] DRD2 Anxiety Disorder 79 prochlorperazine [Dopamine D2 receptor antagonist], trifluoperazine hydrochloride [D2-like dopamine receptor antagonist] ADRB2 Atrial Fibrillation 80 propafenone hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Ventricular Arrhythmia 81 propafenone hydrochloride [Beta-2 adrenergic receptor antagonist], sotalol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Cardiac Arrhythmia 82 propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Coronary Atherosclerosis 82 propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Migraine Disorder 82 propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] ADRB2 Wolff-Parkinson-White Syndrome 82 propranolol hydrochloride [Beta-2 adrenergic receptor antagonist] DRD2 Bipolar Ii Disorder 83 quetiapine fumarate [Dopamine D2 receptor antagonist] HTR2A Bipolar Ii Disorder 84 quetiapine fumarate [Serotonin 2a (5-HT2a) receptor antagonist] PDE4D Chronic Obstructive Pulmonary Disease 85 roflumilast [Phosphodiesterase 4 inhibitor] PDE4D Chronic Bronchitis 86 roflumilast [Phosphodiesterase 4 inhibitor], theophylline [Phosphodiesterase 4 inhibitor] ADRB2 Bronchitis 87 terbutaline sulfate [Beta-2 adrenergic receptor agonist] ADRB2 Ocular Hypertension 88 timolol [Beta-2 adrenergic receptor antagonist], timolol maleate [Beta-2 adrenergic receptor antagonist] HTR2A Anxiety Disorder 89 trifluoperazine hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] CACNA1S Cardiac Arrhythmia 90 verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1F Cardiac Arrhythmia 90 verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1D Cardiac Arrhythmia 90 verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] CACNA1C Cardiac Arrhythmia 90 verapamil hydrochloride [Voltage-gated L-type calcium channel blocker] DRD2 Cardiac Arrhythmia 91 ziprasidone hydrochloride [Dopamine D2 receptor antagonist] DRD2 Ventricular Tachycardia 91 ziprasidone hydrochloride [Dopamine D2 receptor antagonist] HTR2A Cardiac Arrhythmia 92 ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist] HTR2A Ventricular Tachycardia 92 ziprasidone hydrochloride [Serotonin 2a (5-HT2a) receptor antagonist]